Author: Slauta Alexander - sports nutrition specialist and gym trainer | more details >> Graduated from: Belarusian State Pedagogical University named after M. Tank. Specialty: social work, pedagogy. Courses on health-improving fitness and bodybuilding at the Belarusian State University of Physical Culture, at the department of health-improving physical culture. Master of Masters in arm wrestling, 1st adult category in hand-to-hand combat. Prize-winner of the Cup of the Republic of Belarus in hand-to-hand combat. Prize-winner of the Republican Dynamyade in hand-to-hand combat.
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Clenbuterol is a rather interesting drug that has bronchilitis properties. Prescribed for people suffering from asthma. The drug quickly came into bodybuilding and fitness, manifesting itself as an anti-catabolic and fat burner. It is also worth mentioning the increased muscle contraction when taking the drug. Agree, a very necessary set for an athlete, especially during a calorie deficit. Let's look at it in more detail.
Properties and Features
Clenbuterol is used in medicine to widen the airways and reduce shortness of breath. Works as a beta-2 agonist, similar to ephedrine. When you take it:
- Release of fatty acids.
- Adipose tissue is reduced by increasing the production of adrenaline.
- The person's temperature rises.
- Metabolism accelerates.
- Appetite decreases.
- The production of the catabolic hormone cortisol is suppressed. That is, it helps prevent muscle breakdown.
In addition, it has weak anabolic properties. But this is less pronounced than fat burning and its anti-catabolic properties.
Overall, clenbuterol helps you burn fat while keeping your muscles from breaking down. The perfect combination for drying!
Application in strength sports
The drug is actively used in fitness and bodybuilding. Many people take it even if they are not active athletes. Typically, the purpose of such use is weight loss. Clenbuterol is very popular among “phytonies”.
Its main application is:
1. Pre-competition preparation for athletes who aim to preserve the accumulated muscle mass as much as possible, with a low-carbohydrate diet, and also reduce the amount of subcutaneous fat.
2. After completing a course of AS (anabolic steroids) to inhibit the catabolic phase and maintain strength indicators. Since the drug is able to reduce the production of cortisol, it prevents the processes of protein breakdown and the breakdown of glycogen (polysaccharide) stored in muscle cells into glucose. What makes the drug indispensable after a cycle for preserving muscle mass.
3. Improving the quality of training. I assume by quality an improved blood supply to the muscles and an increase in strength indicators. A small dose of clenbuterol before training (20-40 mcg) will give excellent results when using pumping.
10 mcg = 0.01 mg (manufacturers indicate the dosage differently).
Clenbuterol. Deadly fat burner
Clenbuterol is a non-steroidal drug that stimulates β2-adrenergic receptors, which has a bronchodilator effect, promotes bronchial relaxation, and thins sputum. Its main purpose is the treatment of bronchial asthma and chronic obstructive pulmonary disease.
We could end the article with this definition, because... it is written in black and white why this medication is used and by whom. However, not all so simple. Jocks, of course, for the most part are not the smartest people, but even among them there are savvy nuggets with a flexible intellect.
And then one day one of the fans of “iron” sports, and maybe some marathon runner from the Olympic reserve, realized that this common adrenergic agonist can be used not only for clearing the lungs and stimulating the bronchi, but also for effective fat burning in pre-competition preparation .
Attention! The channel's editors do not support the use of medications and potent substances. The publication is for informational purposes only. Before undergoing a course of treatment, you must consult a doctor.
To clarify the pharmacological capabilities of clenbuterol, we present some data from the medical reference book.
As a beta-2 agonist, clenbuterol acts as a fat burner by binding to type 2 beta receptors in adipose and muscle tissue of the human body.
After clenbuterol binds to the receptor, a cascade of biochemical reactions is launched that lead to an increase in the synthesis of cAMP (cyclic adenosine monophosphate). cAMP, in turn, activates enzymes that mobilize fatty acids from adipocytes (fat tissue cells).
In general, the drug has a simple and understandable effect on the body. But let's continue..
The action of clenbuterol on beta-2-adrenergic receptors of the presynaptic membrane increases the release of norepinephrine and adrenaline, which have a powerful fat-burning effect.
Clenbuterol increases the level of basal metabolism by 20-30% of the initial level.
Clenbuterol inhibits the activity of lipoprotein lipase, as a result of which fat deposition in adipose tissue becomes difficult.
Acting on beta-2 adrenergic receptors of the central nervous system, this drug enhances the secretion of thyroid hormones - the body's natural fat burners.
Also, thanks to the stupidity of some consumers and specialists, a huge number of myths and misconceptions have developed around clenbuterol. The main misconception is the complete safety and high effectiveness of this drug.
Let's look at other myths and clarify the effectiveness of the drug clenbuterol:
1) It is not anti-catabolic, as was commonly believed in the 90s and early 2000s;
2) Not suitable for use on PCT, because will very successfully waste all course efforts;
3) Increases cortisol synthesis;
4) It is a stimulator of β2-adrenergic receptors, which triggers the release of catecholamines, norepinephrine and adrenaline, which are activators of the lipolysis process;
5) By stimulating the receptors of the central nervous system, it can enhance the secretion of thyroid hormones, but the combination of clenbuterol and exogenous thyroxine is considered more effective;
6) Burns not only fat, but also muscle tissue. Therefore, its use becomes most productive when taking anabolic drugs;
7) Is a mild diuretic;
Accelerates liptosis (the process of releasing fatty acids from liposomes);
9) Slightly reduces the body’s ability to store glycogen;
10) Increases thermogenesis and body temperature. It is generally accepted that an increase in body temperature of 1 degree accelerates basal metabolism by 5%;
11) Taking the drug in reasonable dosages can increase the basal metabolic rate by up to 15%;
12) The LPR of the drug is ~3 hours, which means taking the drug 2 times a day;
13) Taking beta-blockers can reduce or completely eliminate the effect of clenbuterol;
14) You should not take the drug less than 6 hours before bedtime;
15) You can stop taking clenbuterol abruptly;
16) The main side effects are hand tremors, headaches and tachycardia. In case of overdose, diarrhea, nausea, cramps, and increased sweating are possible;
17) There is an assumption that long-term use of the drug in high doses can provoke hardening of the walls of the aorta, leading to a loss of their elasticity;
18) With long-term use, cardiac hypertrophy is possible, since maple affects smooth muscle fibers and muscle tissue of the heart;
19) In animal studies, the phenomena of necrosis of cardiac muscle tissue were noted;
20) Contraindicated for people who have suffered a myocardial infarction, have hypertoriosis or cardiomyopathy;
21) It is worth noting that the drug is registered with WADA as a doping, but is not an anabolic steroid or a synthetic androgen.
Conclusion.
In my subjective but rather experienced opinion, clenbuterol is the most unsuccessful drug for combating excess weight, even despite all its conventional advantages.
This medication can turn a cheerful, cheerful fat man into a disabled person. You can have a lot of health problems using clenbuterol for fat loss. I’ll quote one of my bodybuilder friends:
“When I hear the word clenbuterol, I shudder!”
The probability of experiencing some unpleasant side effect from this “safe” adrenergic agonist in the form of poor health, terrible tremors, and a complete inability to think and think analytically at work is too high. And it’s especially scary to think about the possibility of strokes and even heart attacks.
People around you will think that you are an alcoholic when they see your trembling limbs, unable to calmly pour coffee from the brewer - the tremors and muscle spasms are so strong when using high dosages of clenbuterol.
And what’s most unpleasant for men is that you can only walk when you need to while sitting, because... it would simply be impossible to hit a white friend while standing from the clenbuterol shake.
Dosage and duration of use
When taking the drug, you need to pay attention to the dosage. The average daily dosage is 40-160 mcg, cases of taking 200 mcg are not uncommon, but 120 mcg is a completely acceptable dose. There is another interesting property of this drug: it increases the level of fat burning from course to course. Typically, an athlete starts with one tablet per day and then increases the dosage by one tablet daily to achieve the optimal dosage. The main thing to remember is that drug tolerance is individual. Listen to your body.
The drug should be taken for two weeks, followed by a break of 14 days, in order for beta-adrenergic receptors to recover. Otherwise, due to loss of receptor sensitivity, the effectiveness of clenbuterol will begin to decline. It is recommended to take daily, despite the high half-life of more than a day.
Misconceptions about Clenbuterol
There are many myths regarding Clenbuterol. One of the most common misconceptions is that the drug has an anti-catabolic - anabolic effect. It did not appear out of nowhere. This was facilitated by testing with animals. However, even huge dosages of more than 1 milligram administered daily to horses produced a similar effect in some animals and only to a small extent.
Experimental tests of Clenbuterol on animals have nothing to do with the effect of the drug on the human body. A dosage of 1000 mcg (1 mg) can be administered to horses. For humans it is lethal. And even if Clenbuterol has an anabolic effect in large doses, then, unfortunately, for an athlete who uses the drug in small quantities, this does not make any difference. Therefore, taking medication for an anti-catabolic effect does not make any sense.
Clenbuterol acts exclusively as a fat burner and is prescribed for asthma. It does not have any other effects; it is advisable to take it during the drying period. Any other properties attributed to Clenbuterol, if there are any, their influence is negligible and completely invisible to the athlete. As a fat burner, on the contrary, Clenbuterol has proven itself only on the positive side. You should not treat it as a “miracle” remedy that in itself gets rid of fat deposits. It has a fat-burning effect only with well-designed training and nutrition.
The drug speeds up metabolism and helps the body begin to use fat as a source of energy, given that it does not receive enough calories from food. It is also necessary to remember about individual characteristics. A well-designed regimen, training, and diet sometimes do not allow the athlete to fully experience the effects of Clenbuterol. The rationality of taking these tablets during the drying period can only be assessed by constant monitoring of the results achieved. The main thing is, in pursuit of the effect, do not forget about caution.
Along with tablets, Clenbuterol can also be purchased in syrup form. The latter contains sugar. This makes it not the best choice for an athlete. It is better to give preference to tablets.
Side effects
Clenbuterol, like any drug, has side effects. These include:
- Nausea;
- Headache;
- Insomnia;
- Increased excitability;
- Sense of anxiety;
- Heart rate (heart rate) disturbances;
- Increased pressure;
- Tremor (hand shaking).
However, don't worry. As a rule, all side effects disappear after 5-7 days of use. Personally, I noticed almost no side effects when using a dosage of 120 mcg. To reduce side effects and increase the duration of use, clenbuterol is taken together with ketotifen.
Uses with other drugs
1. An excellent combination would be the combined use of clenbuterol at a dosage of 120-160 mcg with metformin (2500 mg). Thus, these drugs manage to enhance each other’s actions. In this case, Clenbuterol helps eliminate the negative properties of metformin, in particular, the feeling of fatigue.
2. Anabolic steroids such as oxandrolone and testosterone also have the ability to enhance the effect of clenbuterol.
3. It is recommended to use the drug together with triiodothyronine only for experienced athletes.
Conclusion
Undoubtedly, clenbuterol is very interesting for fans of strength sports, fitness, bodybuilding, etc. According to the rating, the drug is in worldwide demand, and for good reason. Many position it as an indispensable fat burner, but I would call this property secondary, after all, first of all, it is an anti-catabolic. The drug's ability to burn fat cannot be compared to the use of ephedrine with caffeine. Despite all the side effects that may discourage people who decide to take clenbuterol, it justifies its use and is used quite often during drying. I would call it an indispensable assistant in the fight against cortisol and body fat, while it has mild anabolic properties.
Bodybuilding and clenbuterol
The main feature of clenbuterol for a bodybuilder is that the drug combines the ability to burn fat deposits and promote muscle building. Naturally, the increase will not be as significant as when taking some other medications, and will remain within reason.
Clenbuterol should not be used in competitions, as it helps to activate the body's strength and improves performance. And even despite the fact that this medicine is banned by the World Anti-Doping Organization, a very large number of athletes use it to get rid of excess fat and actively build muscle mass.
Clenbuterol is very popular in bodybuilding. Here are just some of the effects it has on the athlete’s body:
- Getting rid of excess fat;
- Drying muscles;
- Increased body temperature;
- Anabolic effect;
- Weight loss;
- Mobilization of the body's emotional resources;
- Decreased appetite;
- Anti-catabolic effect.
